What is INTEPIRDINE used for?

INTEPIRDINE is being researched for the treatment of Alzheimer disease and dementia.

How does INTEPIRDINE work in the brain?

INTEPIRDINE works as a serotonin 6 (5-HT6) receptor antagonist.

Is INTEPIRDINE approved for use yet?

No, INTEPIRDINE is currently in the clinical trial phase (Phase 3) and is not an approved medication.

What kind of molecule is INTEPIRDINE?

INTEPIRDINE is categorized as a small molecule.

What is the chemical name for GSK-742457?

GSK-742457 is another name for the drug INTEPIRDINE.

Is INTEPIRDINE a natural product?

Yes, INTEPIRDINE is identified as a natural product.

Intepirdine | CAS 607742-69-8 | JJZFWROHYSMCMU

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Serotonin receptor antagonist

INTEPIRDINE (also known as GSK-742457) is a small molecule drug currently being studied in clinical trials. It works by blocking the serotonin 6 (5-HT6) receptor in the body.

How it worksINTEPIRDINE acts as a serotonin 6 (5-HT6) receptor antagonist, which means it blocks the action of serotonin at specific receptors.

Used for

Alzheimer diseaseDementia

Conditions

Alzheimer diseaseDementia

Class

Serotonin receptor antagonistCentral Nervous System

How to take

This drug is currently in Phase 3 clinical trials and is not yet widely available for general use.

Talk to your doctor

Questions to ask

·Is INTEPIRDINE currently available through a clinical trial?
·How does a serotonin 6 receptor antagonist affect my condition?

Educational summary derived from FDA labeling, AI-assisted. Not medical advice — consult a healthcare professional. Updated 2026-04-26.

How to take

Talk to your doctor

Frequently asked questions (6)